Specifications
- Supplier
- MedChemExpress
- Catalog No
- HY-100014
- Product Name
- KDM5A-IN-1
- Description
- KDM5A-IN-1 is a potent, orally bioavailable pan-histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively, and with an EC50 value of 960 nM for PC9 H3K4Me3. KDM5A-IN-1 is significantly less potent against other KDM5B enzymes (1A, 2B, 3B, 4C, 6A, 7B)[1].
- Size
- 5 mg
- Datasheet
- http://file.medchemexpress.com/batch_PDF/HY-100014/KDM5A-IN-1-DataSheet-MedChemExpress.pdf
- Msds
- http://file.medchemexpress.com/batch_PDF/HY-100014/KDM5A-IN-1-SDS-MedChemExpress.pdf
- Application
- Cancer-programmed cell death
- Cas No
- 1905481-36-8
- Isotype
- KDM5
- Target Immunogen
- Histone Demethylase
- Storage
- -20°C, 3 years; 4°C, 2 years (Powder)
- Shipping
- Room Temperature
- Product Type
- Reference compound
- Research Area
- Cancer
- Format
- C15H22N4O2
Documentation
No documentation found.
Publications
No publications found.